Pregled po CROSBI profilu: Goran Kragol (CROSBI Profil: 15378, MBZ: 203461)
Pronađeno 68 radova
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1.Electrochemical approach to new derivatives of 4H- 1,3-benzoxazines and 4H-1,3-benzothiazines with potential affinity for DNA/RNA // 23rd Tetrahedron Symposium / Russel, Angela ; Hu, Jinbo (ur.).
Goteborg: University of Gothenburg, 2023. 62, 1 (poster, međunarodna recenzija, sažetak, znanstveni) -
2.The benzothiazine core as a novel motif for DNA- binding small molecules // Molecules, 28 (2023), 4499, 16 doi:10.3390/molecules28114499 (međunarodna recenzija, članak, znanstveni)
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3.Elektrokemijska sinteza novih derivata 1,3- benztiazinskih i 1,3-benzoksazinskih soli s potencijalnim afinitetom prema DNK/RNK, 2022., diplomski rad, diplomski, Fakultet kemijskog inženjerstva i tehnologije, Zagreb
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4.Unprecedented Epimerization of an Azithromycin Analogue: Synthesis, Structure and Biological Activity of 2′-Dehydroxy-5″-Epi-Azithromycin // Molecules, 27 (2022), 3; 1034, 12 doi:10.3390/molecules27031034 (međunarodna recenzija, članak, znanstveni)
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5.Primjena flow-kemije u makrociklizacijskim reakcijama: rekonstrukcija makrolidnog prstena, 2021., diplomski rad, diplomski, Fakultet kemijskog inženjerstva i tehnologije, Zagreb
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6.Clarithromycin inhibits autophagy in colorectal cancer by regulating the hERG1 potassium channel interaction with PI3K // Cell Death & Disease, 11 (2020), 3; 161, 18 doi:10.1038/s41419-020-2349-8 (međunarodna recenzija, članak, znanstveni)
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7.Seco macrolide compounds
(2020) -
8.Efficient N-demethylation of azithromycin using a modified non-classical Polonovski reaction // EFMC-ISMC 2014 - XXIII International Symposium on Medicinal Chemistry
Lisabon, Portugal, 2014. str. 1-2 (poster, međunarodna recenzija, sažetak, znanstveni) -
9.The design of novel classes of macrolides for neutrophil-dominated inflammatory diseases // Future medicinal chemistry, 6 (2014), 6; 657-674 doi:10.4155/fmc.14.14 (međunarodna recenzija, članak, znanstveni)
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10.Regioselective 2-Imino-1, 3-thiazolidine vs. 2-Imino-1, 3-oxazolidine Formation from the Vicinalsec-Amino Alcohol of Desosamine // European journal of organic chemistry, 2013 (2013), 21; 4666-4673 doi:10.1002/ejoc.201300266 (međunarodna recenzija, članak, znanstveni)
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11.Synthesis of novel adamantyl and homoadamantyl substituted β-hydroxybutyric acids // Molecular diversity, 17 (2013), 4; 817-826 doi:10.1007/s11030-013-9481-7 (međunarodna recenzija, članak, znanstveni)
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12.N'-substituted-2'-O, 3'-N-carbonimidoyl bridged macrolides : novel anti-inflammatory macrolides without antimicrobial activity // Journal of medicinal chemistry, 55 (2012), 13; 6111-6123 doi:10.1021/jm300356u (međunarodna recenzija, članak, znanstveni)
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13.Impact of stereochemistry on the biological activity of novel oleandomycin derivatives // Bioorganic & medicinal chemistry, 20 (2012), 7; 2274-2281 doi:10.1016/j.bmc.2012.02.013 (međunarodna recenzija, članak, znanstveni)
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14.Fluorescently labeled macrolides as a tool for monitoring cellular and tissue distribution of azithromycin // Pharmacological research, 66 (2012), 4; 332-342 doi:10.1016/j.phrs.2012.06.001 (međunarodna recenzija, članak, znanstveni)
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15.Novel desosamine-modified 14- and 15-membered macrolides without antibacterial activity // Bioorganic & medicinal chemistry letters, 22 (2012), 10; 3527-3530 doi:10.1016/j.bmcl.2012.03.076 (međunarodna recenzija, članak, znanstveni)
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16.Novel 9a, 11-bridged azalides : One-pot synthesis of N'-substituted 2-imino-1, 3-oxazolidines condensed to an azalide aglycone // Bioorganic & medicinal chemistry, 19 (2011), 1; 556-566 doi:10.1016/j.bmc.2010.10.061 (međunarodna recenzija, članak, znanstveni)
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17.Novel Tandem Reaction for the Synthesis of N'-Substituted 2-Imino-1, 3-oxazolidines from Vicinal (sec- or tert-)Amino Alcohol of Desosamine // European journal of organic chemistry, 14 (2011), 13; 2507-2518 doi:10.1002/ejoc.201001707 (međunarodna recenzija, članak, znanstveni)
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18.Could LogP be a principal determinant of biological activity in 18-crown-6 ethers? Synthesis of biologically active adamantane-substituted diaza-crowns // European Journal of Medicinal Chemistry, 46 (2011), 8; 3444-3454 doi:10.1016/j.ejmech.2011.05.009 (međunarodna recenzija, članak, znanstveni)
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19.Modeling Cellular Pharmacokinetics of 14- and 15-membered Macrolides with Physicochemical Properties // Journal of medicinal chemistry, 54 (2011), 3; 719-733 doi:10.1021/jm101317f (međunarodna recenzija, članak, znanstveni)
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20.Synthesis and Properties of Macrolones Characterized by Two Ether Bonds in the Linker // Bioorganic & medicinal chemistry, 18 (2010), 17; 6578-6588 doi:10.1016/j.bmc.2010.07.007 (međunarodna recenzija, članak, znanstveni)
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21.Novel cage-functionalized building blocks in peptidomimetic design // AMP2010 - Australia-Croatia workshop on antimicrobial peptides and summer school in biophysics Phd programme
Split, 2010. str. 45-45 (poster, međunarodna recenzija, sažetak, stručni) -
22.Sintetski peptidi s neprirodnim adamantanskim aminokiselinama za uporabu kao protutumorski lijekovi
Hrvatski patentni glasnik 9 (2010) 2467. -
23.Transannular Cyclization with Grignard Reagents: Facile Synthetic Routes to Oxaadamantane and Protoadamantane Derivatives // Synlett, 2008 (2008), 3; 405-409 doi:10.1055/s-2008-1032054 (međunarodna recenzija, članak, znanstveni)
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24.Novel 9a-carbamoyl- and 9a-thiocarbamoyl-3-decladinosyl-6-hydroxy and 6-methoxy derivatives of 15-membered macrolides // Bioorganic & Medicinal Chemistry, 15 (2007), 13; 4498-4510 (međunarodna recenzija, članak, znanstveni)
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25.Transannular cyclization with Grignard reagents: an efficient synthesis of oxaadamantane and protoadamantane derivatives // 15th European Symposium on Organic Chemistry ; ESOC 15
Dublin, 2007. (poster, međunarodna recenzija, sažetak, znanstveni)
