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Pregled bibliografske jedinice broj: 363800

Macrolides with anti-inflammatory activity


Čulić, Ognjen; Bosnar, Martina; Marjanović, Nikola; Jelić, Dubravko; Alihodžić, Sulejman; Vela, vanja; Marušić Ištuk, Zorica; Eraković, Vesna; Bošnjak, Berislav; Hrvačić, Boška et al.
Macrolides with anti-inflammatory activity
(2006)


CROSBI ID: 363800 Za ispravke kontaktirajte CROSBI podršku putem web obrasca

Naslov
Macrolides with anti-inflammatory activity

Autori
Čulić, Ognjen ; Bosnar, Martina ; Marjanović, Nikola ; Jelić, Dubravko ; Alihodžić, Sulejman ; Vela, vanja ; Marušić Ištuk, Zorica ; Eraković, Vesna ; Bošnjak, Berislav ; Hrvačić, Boška ; Tomašković, Marija ; Munić, Vesna ; Ivetić, Vanesa ; Hutinec, Antun ; Kragol, Goran ; Leljak, Marija

Broj patenta
WO 20061087644 A2

Godina
2006

Datum patenta
24.08.2006.

Nositelj prava
Glaxosmithkline istraživački centar Zagreb d.o.o., ,

Sažetak
The present invention relates to novel semi-synthetic macrolides having anti-inflammatory activity. More particu-larly the invention relates to 14- and 15-membered macrolides substituted at 4"-position to their pharmaceutically acceptable derivatives, to processes and intermediates for their preparation, to pharmaceutical composition containing them and to their activity and use in the treatment of inflammatory diseases and conditions in humans and animals, especially those diseases associated 4 with excessive secretion of TNF-a, IL-1, IL-8, IL-2 or IL-5 ; and/or inhibitor of excessive lymphocyte proliferation ; and/or excessive granulocyte degranulation.

Izvorni jezik
Engleski

Znanstvena područja
Kemija, Temeljne medicinske znanosti



POVEZANOST RADA



Citiraj ovu publikaciju:

Čulić, Ognjen; Bosnar, Martina; Marjanović, Nikola; Jelić, Dubravko; Alihodžić, Sulejman; Vela, vanja; Marušić Ištuk, Zorica; Eraković, Vesna; Bošnjak, Berislav; Hrvačić, Boška et al.
Macrolides with anti-inflammatory activity
(2006)
Glaxosmithkline istraživački centar Zagreb d.o.o. (2006) Macrolides with anti-inflammatory activity, WO 20061087644 A2.
@patent{patent, author = {\v{C}uli\'{c}, Ognjen and Bosnar, Martina and Marjanovi\'{c}, Nikola and Jeli\'{c}, Dubravko and Alihod\v{z}i\'{c}, Sulejman and Vela, vanja and Maru\v{s}i\'{c} I\v{s}tuk, Zorica and Erakovi\'{c}, Vesna and Bo\v{s}njak, Berislav and Hrva\v{c}i\'{c}, Bo\v{s}ka and Toma\v{s}kovi\'{c}, Marija and Muni\'{c}, Vesna and Iveti\'{c}, Vanesa and Hutinec, Antun and Kragol, Goran and Leljak, Marija}, year = {2006}, keywords = {}, title = {Macrolides with anti-inflammatory activity}, keyword = {} }
@patent{patent, author = {\v{C}uli\'{c}, Ognjen and Bosnar, Martina and Marjanovi\'{c}, Nikola and Jeli\'{c}, Dubravko and Alihod\v{z}i\'{c}, Sulejman and Vela, vanja and Maru\v{s}i\'{c} I\v{s}tuk, Zorica and Erakovi\'{c}, Vesna and Bo\v{s}njak, Berislav and Hrva\v{c}i\'{c}, Bo\v{s}ka and Toma\v{s}kovi\'{c}, Marija and Muni\'{c}, Vesna and Iveti\'{c}, Vanesa and Hutinec, Antun and Kragol, Goran and Leljak, Marija}, year = {2006}, keywords = {}, title = {Macrolides with anti-inflammatory activity}, keyword = {} }




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