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Procjena učinkovitosti i toksičnosti biološki aktivnih tvari
suradnik
Analiza interakcija butirilkolinesteraze s novim inhibitorima i reaktivatorima
suradnik
Analiza interakcija organofosfornih spojeva s esterazama i mogućim metama terapije kod otrovanja
suradnik
Dizajn, sinteza i evaluacija novih protuotrova kod trovanja živčanim bojnim otrovima i pesticidima
suradnik
Naziv
Akcije
Kovarik, Zrinka; Kolić, Dora; Čadež, Tena; Maček Hrvat, Nikolina; Šinko, Goran
Challenging the universality of standard oximes in reactivation of AChE and BChE inhibited by nerve agents // 18 Medical Chemical Defense Conference "Recent Advances - ongoing Challenges" : Book of abstracts. Munich: Bundeswehr Institute of Phramacology and Toxicology, 2023. str. 144-144
Šinko, Goran
Modeling of a near-attack conformation of oxime in phosphorylated acetylcholinesterase via a reactivation product, a phosphorylated oxime // Chemico-biological interactions, 383 (2023), 110656, 9. doi: 10.1016/j.cbi.2023.110656
Kolić, Dora; Spahić, Zlatan; Šinko, Goran; Primožič, Ines; Kovarik, Zrinka
Novel imidazolium oximes as potent reactivators of organophosphate-inhibited human butyrylcholinesterase // FEBS Open Bio, 13, S2. 2023. str. 206-206 doi: 10.1002/2211-5463
Pehar, Vesna ; Kolić, Dora ; Zandona, Antonio ; Šinko, Goran ; Katalinić, Maja ; Stepanić, Višnja ; Kovarik, Zrinka
Selected herbicides screened for toxicity and analysed as inhibitors of both cholinesterases // Chemico-biological interactions, 379 (2023), 110506, 13. doi: 10.1016/j.cbi.2023.110506
Šinko, Goran
50. godišnjica osnutka baze struktura bioloških makromolekula // Kemija u industriji : časopis kemičara i tehnologa Hrvatske, 72 (2023), 1-2; 95-101. doi: 10.15255/KUI.2022.029
Kovarik, Zrinka ; Čadež, Tena ; Kolić, Dora ; Šinko, Goran
Assessment of four organophosphorus pesticides as inhibitors of human cholinesterases // 17th International Symposium on Cholinergic Mechanisms (ISCM2022) : Programme and Abstracts / Kovarik, Zrinka ; Primožič, Ines (ur.). Zagreb: Institut za medicinska istraživanja i medicinu rada, 2022. str. 45-45
Šinko, Goran
Modeling of a Michaelis type complex between phosphorylated acetylcholinesterase and an oxime via a reactivation product the phosphorylated oxime // 14th International Meeting on Cholinesterases-8th International Conference on Paraoxonases Abstract Book / Lamba, Doriano ; Bolognesi, Maria Laura (ur.). Bolonja, 2022. str. 43-43
Miličević, Ante ; Šinko, Goran
Use of connectivity index and simple topological parameters for estimating the inhibition potency of acetylcholinesterase // SAUDI PHARMACEUTICAL JOURNAL, 30 (2022), 4; 369-376. doi: 10.1016/j.jsps.2022.01.025
Miličević, Ante ; Šinko, Goran
Evaluation of the key structural features of various butyrylcholinesterase inhibitors using simple molecular descriptors // Molecules, 27 (2022), 6894, 11. doi: 10.3390/molecules27206894
Kolić, Dora ; Šinko, Goran ; Jean, Ludovic ; Chioua, Mourad ; Dias, José ; Marco-Contelles, José ; Kovarik, Zrinka
Cholesterol oxime olesoxime (TRO19622) as a potential reactivator of nerve agent-inhibited cholinesterases // FEBS Open Bio. 2022. str. 132-132 doi: 10.1002/2211-5463.13440