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Transcriptional expression and functional activity of mu-opioid receptors (MOR) on myelo-monocytic HL-60 cell line (CROSBI ID 535406)

Prilog sa skupa u zborniku | izvorni znanstveni rad | međunarodna recenzija

Gabrilovac, Jelka ; Breljak, Davorka ; Čupić, Barbara Transcriptional expression and functional activity of mu-opioid receptors (MOR) on myelo-monocytic HL-60 cell line // 8th International Congress of Neuroimmunology Free Papers / Takashi, Tabira ; Takashi, Yamamura ; Junichi, Kira (ur.). Bolonja: Monduzzi Editore S.p.A. - Medimond Inc., International Proceedings Division, 2007. str. 287-292

Podaci o odgovornosti

Gabrilovac, Jelka ; Breljak, Davorka ; Čupić, Barbara

engleski

Transcriptional expression and functional activity of mu-opioid receptors (MOR) on myelo-monocytic HL-60 cell line

Opioid receptors, highly expressed on cells of central nervous system, were also found on cells of hematopoietic origin, but at much lower density. In this study we have examined transcriptional expression of mu-opioid receptors (MOR) on HL-60 cells of myelo-monocytic origin, at their basal state. Functionality of the MOR on these cells was examined by following Ca++ mobilization triggered by selective agonist of alkaloid (morphine) and peptide (endomorphin-2) structure. The data obtained have shown that cells of myelo-monocytic HL-60 line, at their basal state, express MOR both at the level of mRNA and at the level of a functionally active protein capable of transmitting intracellular signals via Ca++ upon ligation with selective agonists of alkaloid or peptide structure.

mu-opioid receptors ; transcriptional expression ; functional activity ; morphine ; endomorphin-2

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Podaci o prilogu

287-292.

2007.

objavljeno

Podaci o matičnoj publikaciji

8th International Congress of Neuroimmunology Free Papers

Takashi, Tabira ; Takashi, Yamamura ; Junichi, Kira

Bolonja: Monduzzi Editore S.p.A. - Medimond Inc., International Proceedings Division

978-88-7587-324-0

7891-352X

Podaci o skupu

Nepoznat skup

predavanje

29.02.1904-29.02.2096

Povezanost rada

Temeljne medicinske znanosti